Jakupec, Michael A.

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Journal Article

Mendoza-Ferri, Maria G.; Hartinger, Christian G.; Mendoza, Marco A.; Grössl, Michael; Egger, Alexander E.; Eichinger, Rene E.; Mangrum, John B.; Farrell, Nicholas P.; Maruszak, Magdalena; Bednarski, Patrick J.; Klein, Franz; Jakupec, Michael A.; Nazarov, Alexey A.; Severin, Kay; Keppler, Bernhard K. (2009). Transferring the Concept of Multinuclearity to Ruthenium Complexes for Improvement of Anticancer Activity. Journal of medicinal chemistry, 52(4), pp. 916-925. American Chemical Society 10.1021/jm8013234

Biba, Florian; Grössl, Michael; Egger, Alexander; Jakupec, Michael A.; Keppler, Bernhard K. (2009). A Novel Cytotoxic Cerium Complex: Aquatrichloridobis(1,10-phenanthroline)cerium(III) (KP776). Synthesis, Characterization, Behavior in H2O, Binding towards Biomolecules, and Antiproliferative Activity. Chemistry & Biodiversity, 6(12), pp. 2153-2165. Verlag Helvetica Chimica Acta 10.1002/cbdv.200900011

Hartinger, Christian G.; Jakupec, Michael A.; Zorbas-Seifried, Stefanie; Grössl, Michael; Egger, Alexander; Berger, Walter; Zorbas, Haralabos; Dyson, Paul J.; Keppler, Bernhard K. (2008). KP1019, A New Redox-Active Anticancer Agent - Preclinical Development and Results of a Clinical Phase I Study in Tumor Patients. Chemistry & Biodiversity, 5(10), pp. 2140-2155. Verlag Helvetica Chimica Acta 10.1002/cbdv.200890195

Berger, Isabella; Hanif, Muhammad; Nazarov, Alexey A.; Hartinger, Christian G.; John, Roland O.; Kuznetsov, Maxim L.; Grössl, Michael; Schmitt, Frederic; Zava, Olivier; Biba, Florian; Arion, Vladimir B.; Galanski, Markus; Jakupec, Michael A.; Juillerat-Jeanneret, Lucienne; Dyson, Paul J.; Keppler, Bernhard K. (2008). In Vitro Anticancer Activity and Biologically Relevant Metabolization of Organometallic Ruthenium Complexes with Carbohydrate-Based Ligands. Chemistry - a European journal, 14(29), pp. 9046-9057. Wiley-VCH 10.1002/chem.200801032

Grössl, Michael; Reisner, Erwin; Hartinger, Christian G.; Eichinger, Rene; Semenova, Olga; Timerbaev, Andrei R.; Jakupec, Michael A.; Arion, Vladimir B.; Keppler, Bernhard K. (2007). Structure−Activity Relationships for NAMI-A-type Complexes (HL)[ trans -RuCl 4 L( S -dmso)ruthenate(III)] (L = Imidazole, Indazole, 1,2,4-Triazole, 4-Amino-1,2,4-triazole, and 1-Methyl-1,2,4-triazole): Aquation, Redox Properties, Protein Binding, and Antiproliferative Activity. Journal of medicinal chemistry, 50(9), pp. 2185-2193. American Chemical Society 10.1021/jm061081y

Berger, Isabella; Nazarov, Alexey A.; Hartinger, Christian G.; Grössl, Michael; Valiahdi, Seied-M.; Jakupec, Michael A.; Keppler, Bernhard K. (2007). A glucose derivative as natural alternative to the cyclohexane-1,2-diamine ligand in the anticancer drug oxaliplatin? ChemMedChem, 2(4), pp. 505-514. Wiley-VCH 10.1002/cmdc.200600279

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